Synonym(s):

CAS Number

136194-77-9

Commodity Code

2933998090

MDL Number

MFCD00236434

Notes

Novel, very potent PKC inhibitor with high selectivity for the A-group of PKC isotypes (alpha, beta, and gamma), with IC50 values in the 2-10 nM range.  Little or no inhibition of the B- and C-groups of PKC isotypes, even at much higher concentrations.    Bioorg. Med. Chem. Lett. 3:  1959-1964 (1993).